Compile Data Set for Download or QSAR
maximum 50k data
Found 20 of non-affinity data for polymerid = 1024,2148
TargetAromatase(Homo sapiens (Human))
Tohoku Pharmaceutical University

LigandPNGBDBM9991((2S,6S,15S)-6-hydroxy-2-(methoxymethyl)-15-methylt...)
Affinity DatapH: 7.5 T: 2°CAssay Description:The enzyme activity was assayed by measuring the 3H-labeled H2O formed from [1beta-3H] Androstenedione during aromatization. After incubation, the re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku Pharmaceutical University

LigandPNGBDBM24303((2-methoxy-4-{[3-methoxy-4-(sulfamoyloxy)phenyl](1...)
Affinity DatapH: 7.5 T: 2°CAssay Description:The extent of in vitro inhibition of aromatase activities was assessed using intact monolayers of JEG-3 cells. Aromatase activity was measured using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku Pharmaceutical University

LigandPNGBDBM8939(4-(5-Methoxy-7b-methyl-3,7b-dihydro-2H-1-oxa-cyclo...)
Affinity DataAssay Description:The enzyme activity was assayed by measuring the 3H-labeled H2O formed from [1beta-3H]androstenedione during aromatization. After incubation, the rea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku Pharmaceutical University

LigandPNGBDBM8947(6,7-Dihydroxy-2-(1H-imidazol-5-ylmethyl)-3,4-dihyd...)
Affinity DataAssay Description:The enzyme activity was assayed by measuring the 3H-labeled H2O formed from [1beta-3H]androstenedione during aromatization. After incubation, the rea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku Pharmaceutical University

LigandPNGBDBM8948(1-{[4-(3-methoxyphenyl)phenyl]methyl}-1H-imidazole...)
Affinity DataAssay Description:The enzyme activity was assayed by measuring the 3H-labeled H2O formed from [1beta-3H]androstenedione during aromatization. After incubation, the rea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku Pharmaceutical University

LigandPNGBDBM8949(3-[4-(1H-imidazol-1-ylmethyl)phenyl]phenol | BW95 ...)
Affinity DataAssay Description:The enzyme activity was assayed by measuring the 3H-labeled H2O formed from [1beta-3H]androstenedione during aromatization. After incubation, the rea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku Pharmaceutical University

LigandPNGBDBM8950(2-[4-(1H-imidazol-1-ylmethyl)phenyl]benzene-1,4-di...)
Affinity DataAssay Description:The enzyme activity was assayed by measuring the 3H-labeled H2O formed from [1beta-3H]androstenedione during aromatization. After incubation, the rea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku Pharmaceutical University

LigandPNGBDBM8952(4-Imidazol-1-ylmethyl-biphenyl-2,3,4-triol | 4-[4-...)
Affinity DataAssay Description:The enzyme activity was assayed by measuring the 3H-labeled H2O formed from [1beta-3H]androstenedione during aromatization. After incubation, the rea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku Pharmaceutical University

LigandPNGBDBM8954(1-[(2,5-dimethoxy-1,1-biphenyl-4-yl)methyl]-1H-imi...)
Affinity DataAssay Description:The enzyme activity was assayed by measuring the 3H-labeled H2O formed from [1beta-3H]androstenedione during aromatization. After incubation, the rea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku Pharmaceutical University

LigandPNGBDBM8955(1-[(3,4-dimethoxy-1,1-biphenyl-4-yl)methyl]-1H-imi...)
Affinity DataAssay Description:The enzyme activity was assayed by measuring the 3H-labeled H2O formed from [1beta-3H]androstenedione during aromatization. After incubation, the rea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku Pharmaceutical University

LigandPNGBDBM8957(1-[(3,4,5-trimethoxy-1,1-biphenyl-4-yl)methyl]-1H-...)
Affinity DataAssay Description:The enzyme activity was assayed by measuring the 3H-labeled H2O formed from [1beta-3H]androstenedione during aromatization. After incubation, the rea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku Pharmaceutical University

LigandPNGBDBM9466(4-(9-Phenyl-9H-fluoren-9-yl)-4H-1,2,4-triazole | F...)
Affinity DatapH: 7.4 T: 2°CAssay Description:The enzyme activity was assayed by measuring the 3H-labeled H2O formed from [1beta, 2beta-3H] testosterone or [1beta-3H] androstenedione during aroma...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku Pharmaceutical University

LigandPNGBDBM9467(1-(9-Phenyl-9H-fluoren-9-yl)-1H-1,2,3-triazole | F...)
Affinity DatapH: 7.4 T: 2°CAssay Description:The enzyme activity was assayed by measuring the 3H-labeled H2O formed from [1beta, 2beta-3H] testosterone or [1beta-3H] androstenedione during aroma...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku Pharmaceutical University

LigandPNGBDBM9474(4-[2-(1H-Imidazol-1-yl)ethoxy]-7-methoxy-2H-chrome...)
Affinity DatapH: 7.4 T: 2°CAssay Description:The enzyme activity was assayed by measuring the 3H-labeled H2O formed from [1beta, 2beta-3H] testosterone or [1beta-3H] androstenedione during aroma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku Pharmaceutical University

LigandPNGBDBM9479(7-(1H-1,2,4-Triazol-1-ylmethyl)-2H-chromen-2-one |...)
Affinity DatapH: 7.4 T: 2°CAssay Description:The enzyme activity was assayed by measuring the 3H-labeled H2O formed from [1beta, 2beta-3H] testosterone or [1beta-3H] androstenedione during aroma...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku Pharmaceutical University

LigandPNGBDBM9480(7-[2-(1H-Imidazol-1-yl)ethoxy]-2H-chromen-2-one | ...)
Affinity DatapH: 7.4 T: 2°CAssay Description:The enzyme activity was assayed by measuring the 3H-labeled H2O formed from [1beta, 2beta-3H] testosterone or [1beta-3H] androstenedione during aroma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku Pharmaceutical University

LigandPNGBDBM9481(8-(1H-Imidazol-1-ylmethyl)-7-methoxy-2H-chromen-2-...)
Affinity DatapH: 7.4 T: 2°CAssay Description:The enzyme activity was assayed by measuring the 3H-labeled H2O formed from [1beta, 2beta-3H] testosterone or [1beta-3H] androstenedione during aroma...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku Pharmaceutical University

LigandPNGBDBM9484(7-methoxy-4-(pyridin-4-yl)-2H-chromen-2-one | Coum...)
Affinity DatapH: 7.4 T: 2°CAssay Description:The enzyme activity was assayed by measuring the 3H-labeled H2O formed from [1beta, 2beta-3H] testosterone or [1beta-3H] androstenedione during aroma...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku Pharmaceutical University

LigandPNGBDBM24302((2-methoxy-5-{[4-methoxy-3-(sulfamoyloxy)phenyl](1...)
Affinity DatapH: 7.5 T: 2°CAssay Description:The extent of in vitro inhibition of aromatase activities was assessed using intact monolayers of JEG-3 cells. Aromatase activity was measured using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku Pharmaceutical University

LigandPNGBDBM8938(7-(1H-Imidazol-5-ylmethyl)-8-methyl-5,6-dihydro-na...)
Affinity DataAssay Description:The enzyme activity was assayed by measuring the 3H-labeled H2O formed from [1beta-3H]androstenedione during aromatization. After incubation, the rea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed